N137745-50mgNelfinavir Mesylate
面议
- 阿拉丁
- 生产商
- N137745-50mg
- 现货
- 全国
规格 |
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耗材描述
属性
存贮条件 | 储存温度2-8℃ |
描述
应用 | An antiviral. HIV protease inhibitor. |
产品介绍 | Nelfinavir Mesylate 是强效的HIV protease抑制剂,Ki为2 nM。 |
生化机理 | Nelfinavir is an orally bioavailable inhibitor of the HIV-1 protease (Ki =2 nM) that is used in combination with HIV reverse transcriptase inhibitors for the treatment of HIV infection. Nelfinavir demonstrates anti-cancer activity, selectively preventing the growth of HER2-positive breast cancer cells in vitro by inhibiting Hsp90 (IC50 = 3.1 μM). |
别名 | 甲磺酸奈非那韦; 2-[(2R,3R)-2-羟基-3-[(3-羟基-2-甲基苯甲酰)氨基]-4-(苯基硫)丁基]-(3S,4aS,8aS)-N-叔丁基十氢异喹啉-3-甲酰胺甲磺酸盐;(3S,4aS,8aS)-N-(1,1-Dimethylethyl)decahydro-2-[(2R,3R)-2-hydroxy-3-[(3-hydroxy-2-methylbenzoyl)amino]-4-(phenylthio)butyl]-3-isoquinolinecarboxamide mesylate |
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