耗材描述

• 分子式 C₂₅H₃₄N₄O₂ · C₄H₄O₄
• 分子量538.64
• Beilstein号
• EC号
• MDL号 MFCD01321056
• PubChem编号 24278113

属性

描述

应用	WAY-100635 maleate salt has been used as a 5-HT1A serotonin receptor antagonist: · to study whether the behavior of the cleaner wrasse is regulated by serotonin activity · to block activity of 3,4 methylenedioxymethamphetamine (MDMA) used to induce oxytocin release in male Wistar rats to increase their social behavior · to study the role of serotonin during metamorphosis of the ascidian Phallusia mammillata larvae
产品介绍	WAY-100635马来酸盐是5-HT受体拮抗剂，IC50为0.95nM
生化机理	WAY-100635 maleate salt is a potent, selective and high affinity SR-2B antagonist with a pIC50 of 10.4. The affinity (pKi) of WAY-100635 maleate salt for tSR-2B is 9.5. In addition, WAY-100635 maleate salt also blocks serotonin-evoked contraction of rat isolated stomach fundus.
别名	N- [2- [4-（2-甲氧基苯基）-1-哌嗪基] 乙基]-N-2-吡啶基环己基甲酰胺 马来酸盐;N-[2-[4-(2-Methoxyphenyl)-1-piperazinyl]ethyl]-N-2-pyridinylcyclohexanecarboxamide maleate salt

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