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CAS No. : 1254035-84-1
MCE 国际站:AZD1979
产品活性:AZD1979 是一个 Melanin-concentrating hormone receptor 1 (MCHr1) 拮抗剂, 其 IC50 值约为 12 nM。
研究领域:GPCR/G Protein | Neuronal Signaling
作用靶点:MCHR1 (GPR24)
In Vivo: In DIO mice, initial AZD1979-mediate body weight loss is driven by decreasing food intake, but an additional component of preserving energy expenditure is apparent in pair-feeding and indirect calorimetry studies. AZD1979 also dose-dependently reduces body weight in dogs.
相关产品:Clinical Compound Library Plus | Bioactive Compound Library Plus | GPCR/G Protein Compound Library | Neuronal Signaling Compound Library | Clinical Compound Library | Endocrinology Compound Library | Anti-Obesity Compound Library | Heterocyclic Compound Library | Membrane Protein-targeted Compound Library | Membrane Receptor-targeted Compound Library | GW-803430 | hMCH-1R antagonist 1 | MCH(human, mouse, rat) TFA | SB-568849 | SNAP 94847 hydrochloride | MCHR1 antagonist 3 | ATC0175 | MCHR1 antagonist 1 | Ac-hMCH(6-16)-NH2 | MCH-1 antagonist 1 | MCHR1 antagonist 2 | TC-MCH 7c | (Phe13,Tyr19)-MCH (human, mouse, rat) | Neuropeptide EI, rat | BMS-819881 | Melanin Concentrating Hormone, salmon TFA | [Ala17]-MCH | ALB-127158(a) | BMS-814580 | NGD-4715 | Ethyl linolenate
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