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CAS No. : 522606-67-3
MCE 国际站:SID 3712249
产品活性:SID 3712249 (MiR-544 Inhibitor 1) 是一种 miR-544 生物合成抑制剂。SID 3712249 直接与前体 miRNA 结合。SID 3712249 阻断成熟 microRNA 的产生并减少 miR-544、HIF-1α 和 ATM 转录物。SID 3712249 可用于癌症研究。
研究领域:Epigenetics | Apoptosis
作用靶点:MicroRNA | Apoptosis
In Vitro: SID 3712249 (compound 1, 20 nM, 48 h) disrupts miR-544-mediated inhibition of BMI1 based on significant increases in the RFP/BFP ratio.
SID 3712249 (20 nM, 48 h) inhibits precursor but not mature miR-544 binding to BMI1 or mTOR3’-UTR.
SID 3712249 (20 nM, 48 h) results in accumulation of pre-miR-544 and a decrease in miR-544 levels in MCF10A cells.
SID 3712249 (20 nM, 5 days) induces apoptosis in MDA-MB-231 and MCF- 7 cells and has no effect on cell survival in normoxic conditions.
In Vivo: SID 3712249 (compound 1, 100 μL of 40 μM, intraperitoneal injection) inhibited tumor growth in MDA-MB-231-GFP-luc tumor model.
SID 3712249 (20 nM, pre-treated GFP-labeled MDA-MB-231 cells, intraperitoneal injection) inhibited tumor growth in MDA-MB-231-GFP-luc tumor model.
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