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CAS No. : 58-46-8
MCE 国际站:Tetrabenazine
产品活性:Tetrabenazine (Ro 1-9569) 是一种可逆的囊泡单胺转运蛋白 VMAT2 位点抑制剂,其 Kd 值为 1.34 nM,可用于亨廷顿舞蹈病等多动性运动障碍相关疾病研究。
研究领域:Membrane Transporter/Ion Channel
作用靶点:Monoamine Transporter
In Vivo: Tetrabenazine (subcutaneous injection, 1-10 mg/kg, once) can reduce the aggressive behavior in a dose-dependent manner and the levels of neurotransmitter molecules NE, DA and 5-HT in adult male mice.Tetrabenazine (intraperitoneal injection, 0-2 mg/kg, once) has selective effects on movement which can significantly attenuate morphine-induced hypermobility but oral tremors and stereotyped behaviors in male ICR mice.Tetrabenazine (intraperitoneal injection, 0.25-2 mg/kg, once a week) increases tremulous jaw movement (TJM) in a dose-dependent manner in adult male Sprague-Dawley rat.
相关产品:Drug Repurposing Compound Library Plus | FDA-Approved Drug Library Plus | FDA-Approved Drug Library Mini | Bioactive Compound Library Plus | Membrane Transporter/Ion Channel Compound Library | FDA-Approved Drug Library | CNS-Penetrant Compound Library | Peptidomimetic Library | Drug Repurposing Compound Library | Orally Active Compound Library | FDA Approved & Pharmacopeial Drug Library | Drug-Induced Liver Injury (DILI) Compound Library | Targeted Diversity Library | Rare Diseases Drug Library | Human Metabolite Library | Heterocyclic Compound Library | Off-patent Drug Library | Membrane Protein-targeted Compound Library | Membrane Receptor-targeted Compound Library | Cysteine Targeted Covalent Library | Tetrabenazine Racemate | FFN511 | Cavα2δ1&NET-IN-1 | Nisoxetine | Tetrabenazine Metabolite | Trans (2,3)-Dihydrotetrabenazine | Cavα2δ1&NET-IN-2 | (+)-Tetrabenazine-d6 | hENT4-IN-1 | Reserpine-d9 | GZ-793A | Radafaxine hydrochloride | Reserpine | Valbenazine | FFN200 dihydrochloride | Tetrabenazine mesylate | Vanilpyruvic acid | VMAT2-IN-2 tosylate | 13-Hydroxyisobakuchiol | Pseudoisocyanine iodide
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