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CAS No. : 1902954-60-2
MCE 国际站:Abeprazan
产品活性:Abeprazan (DWP14012) 是一种钾竞争性酸 (potassium-competitive acid) 阻滞剂。Abeprazan 通过可逆的钾竞争性离子结合抑制 H+,K+- ATPase,而无需酸激活。Abeprazan 是一种潜在的质子泵抑制剂,用于研究与酸相关的疾病。
研究领域:Membrane Transporter/Ion Channel
作用靶点:Proton Pump
In Vitro: The mechanism of action of Abeprazan is reversibly binding to H+, K+‐ATPase, and, unlike that of PPIs, does not require acidic environment for drug activation.
In Vivo: Abeprazan inhibits acid secretion in a dose-dependent manner and the inhibition of gastric acid secretion was equal to or greater than that of vonoprazan, a previously approved P-CAB, in various in vivo studies using pylorus-ligated rats, lumen-perfused rat models and heidenhain pouch dog models.
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