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CAS No. : 1372206-64-8
MCE 国际站:THX-B
产品活性:THX-B 是一种有效的、非多肽类型的 p75NTR (神经营养蛋白受体 p75) 拮抗剂。THX-B 可用于糖尿病、肾病、神经退行性和炎症性疾病的研究。
研究领域:GPCR/G Protein | Neuronal Signaling
作用靶点:Neurotensin Receptor
In Vitro: THX-B (10 μM, 4 days) decreases proliferation of myoblasts.
THX-B (10 μM, 1 h) inhibits NGF-induced phosphorylation of ERK1/2 in C2C12 myoblasts.
THX-B (20 μM, 24 h) decreases photoreceptor cell death and reactive gliosis in cultured rd10 retinas.
In Vivo: THX-B (50 μg in 125 μL PBS, i.p. weekly for 4 weeks) improves bladder function in a mouse model of diabetic voiding dysfunction.
THX-B (2 μL of 2 μg/μL, IVT injection, a single dose) elicits a neuroprotective effect on photoreceptor cells in P17 rd10 mice.
THX-B (40 μg in 20 μL, IVT injection) resolves the inflammatory, vascular, and neurodegenerative phases of the retinal pathology.
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