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CAS No. : 2470969-89-0
MCE 国际站:SIRT1-IN-2
产品活性:SIRT1-IN-2 (compound 3h) 是一种有效且选择性的 SIRT1 (沉默信息调节因子1)抑制剂,其IC50 为 1.6 μM。
研究领域:Cell Cycle/DNA Damage | Epigenetics
作用靶点:Sirtuin
In Vitro: SIRT1-IN-2 (compound 3h) (0-100 μM, 48 h) inhibits the proliferation of Human cancer cell lines including K562, HCT-116, HepG2, A549, and MCF-7, and shows significantly less cytotoxic on 293T cells and HUVEC.
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