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CAS No. : 113-79-1
MCE 国际站:Argipressin
产品活性:Argipressin (Arg8-vasopressin) 可与血管精氨酸加压素受体 V1、V2 和 V3 结合,其在 A7r5 大鼠主动脉平滑肌细胞中对 V1 的 Kd 值为 1.31 nM。
研究领域:GPCR/G Protein
作用靶点:Vasopressin Receptor
In Vitro: Argipressin binds to the vascular arginine vasopressin receptor, V1, with a Kd value of 1.31 nM in A7r5 rat aortic smooth muscle cells. It also stimulates the intracellular release of calcium in A7r5 cells (EC50=5 nM). AVP-induced [Ca2+]i signals and immunized activity against S-100 in DRG cell culture. The minimum effective concentrations of Argipressin causing [Ca2+]i responses are 100 pM in non-neuronal cells in DRG culture.
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