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CAS No. : 13602-53-4
MCE 国际站:Angiotensin III, human, mouse
产品活性:Angiotensin III, human, mouse 是一种七肽,为血管紧张素 2 型受体 (AT2R) 激动剂,对 AT2R 和 AT1R 的 IC50 值分别为 0.648 nM 和 21.1 nM。
研究领域:GPCR/G Protein
作用靶点:Angiotensin Receptor
In Vitro: Angiotensin III, human, mouse is a heptapeptide, acts as an endogenous angiotensin type 2 receptor (AT2R) agonist, with IC50s of 0.648 nM and 21.1 nM for AT2R and AT1R, respectively.
In Vivo: Angiotensin III (7, 14 and 28 nmol/kg/min) increases urine sodium excretion (UNaV), fractional excretion of sodium (FENa), and fractional excretion of lithium (FELi) in SD rat. In RAS (renin-angiotensin system), Angiotensin III increases sympathetic nerve activity and vasopressin release and decreases the baroreflex leading to higher blood pressure in rats.
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