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CAS No. : 30220-46-3
MCE 国际站:Ingenol
产品活性:Ingenol 是一种 PKC 激活剂,Ki 值为 30 μM,具有抗肿瘤活性。
研究领域:Epigenetics | TGF-beta/Smad
作用靶点:PKC
结构分类:萜类 | 二萜
来源:植物 | 禾本科 | 千金子
In Vitro: Ingenol is a PKC activator, with a Ki of 30 μM. Ingenol induces ornithine decarboxylase activity (1, 3 mM), and causes morphological changes (1 mM) in primary mouse epidermal keratinocytes. Ingenol (125 μM, 250 μM, 500 μM, 1 mM) also inhibits cell-cell communication.
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