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CAS No. : 514-47-6
MCE 国际站:Euphol
产品活性:Euphol 是一种四环三萜醇,是从 Euphorbia tirucalli 的汁液中分离出来的,具有抗炎和免疫调节作用,具有口服活性。 Euphol 通过一种可逆机制抑制单酰基甘油脂肪酶 (MGL) 的活性,IC50=315 nM。 外周 MGL 抑制可调节内源性大麻素系统从而阻止炎症性疼痛的发展。
研究领域:Metabolic Enzyme/Protease
作用靶点:MAGL | Endogenous Metabolite
结构分类:萜类 | 三萜 | 结构分类
来源:植物 | 大戟科 | 绿玉树
In Vitro: Euphol (0.01-0.3 mM; 24-72 hours) markedly inhibits T47D cells proliferation, the IC50 values of euphol treatment for 24, 48 and 72 h were 0.26, 0.22 and 0.13 mM, respectively.Euphol (0.03 mM; 48 or 72 hours) leads to cell cycle arrest by regulating expression of cell cycle-associated proteins.
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