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Khellin

CAS No. : 82-02-0

MCE 国际站：Khellin

产品活性：Khellin 是一种呋喃并色酮，能从 Ammi visnuga L. 中提取得到。Khellin 是一种 EGFR 抑制剂，其 IC₅₀ 为 0.15 µM。Khelline 在体外具有抗增殖活性。Khellin 具有抗痉挛和冠状动脉舒张作用。

研究领域：JAK/STAT Signaling  |  Protein Tyrosine Kinase/RTK

作用靶点：EGFR

结构分类：苯丙素类  |  木脂素

来源：植物  |  唇形科  |  椴叶鼠尾草  |  植物  |  伞形科

In Vitro: Khelline exhibits anti-proliferative activity for MCF-7 cells and Hela cells.
Khellin inhibits the pathways of Ca²⁺ influx which are activated by both noradrenaline and high K⁺.

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