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CAS No. : 1620401-82-2
MCE 国际站:UNC0379
产品活性:UNC0379 是一个选择性的底物竞争性的赖氨酸甲基转移酶 SETD8 (KMT5A) 抑制剂,IC50 值为 7.3 μM,KD 值 of 18.3 μM。UNC0379 可用于炎症癌症的研究,如肺纤维化,卵巢癌,神经母细胞瘤。
研究领域:Epigenetics
作用靶点:Histone Methyltransferase
In Vitro: UNC0379 (1-10 μM, 9 days) inhibits HGSOC cells proliferation.
UNC0379 (10 μM, 96 h) increases in the proportion of sub-G1 phase cells in HGSOC cells.
UNC0379 (10 μM, 48 h) induces myofibroblast de-differentiation and inhibits additional fibroblast to myofibroblast differentiation.
In Vivo: UNC0379 (intratracheal administration, 1 mg/kg/day, on day7, 8, and 9) ameliorates the lung fibrosis in Bleomycin (BLM)-induced lung fibrosis mouse.
相关产品:Bioactive Compound Library Plus | Epigenetics Compound Library | Immunology/Inflammation Compound Library | Histone Modification Research Compound Library | Anti-Cancer Compound Library | Reprogramming Compound Library | Anti-Blood Cancer Compound Library | Targeted Diversity Library | Anti-Pulmonary Fibrosis Compound Library | Heterocyclic Compound Library | Membrane Protein-targeted Compound Library | Highly Selective Inhibitors Library | PRMT5-IN-17 | EZM0414 | BIX-01294 | WDR5-IN-5 | PRMT5-IN-22 | Gambogenic acid | SGC707 | Dot1L-IN-7 | MS1943 | PRMT5-IN-21 | NSD3-IN-3 | DCLX069 | MAK683 | DS-437 | EPZ020411 | WDR5-IN-4 TFA | Amodiaquine dihydrochloride | Furamidine | SMYD3-IN-2 | UNC0642 | Chaetocin | UNC0646 | UNC0224 | EBI-2511 | BVT948 | MM-401 | CMP-5 | EPZ-719
热门产品线:重组蛋白 | 化合物库 | 天然产物 | 荧光染料 | PROTAC | 同位素标记物 | 寡核苷酸 | 抗体 | 点击化学
Trending products:Recombinant Proteins | Bioactive Screening Libraries | Natural Products | Fluorescent Dye | PROTAC | Isotope-Labeled Compounds | Oligonucleotides | Antibodies | Click Chemistry
货号: HY-12335
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