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CAS No. : 2360909-50-6
MCE 国际站:PD-1-IN-24
产品活性:PD-1-IN-24 (compound 1) 是具有口服活性的 PD-1 的抑制剂。
研究领域:Immunology/Inflammation
作用靶点:PD-1/PD-L1
In Vivo: PD-1-IN-24 (compound 1, 15mg/kg, PO, BID) exhibits TGI(%) of 19.96% in the subcutaneous 4T1 murine breast cancer model in BALB/c mice.
PD-1-IN-24 (compound 1, 15mg/kg, PO, BID) dose-dependently inhibits tumor growth in the Bl6F10 models with TGI% of 35.59% (30 mg/kg), 38.87% (60 mg/kg) and 47.35% (120 mg/kg), respectively.
相关产品:Natural Product-like Compound Library | Bioactive Compound Library Plus | Immunology/Inflammation Compound Library | Anti-Cancer Compound Library | Small Molecule Immuno-Oncology Compound Library | Anti-Breast Cancer Compound Library | Anti-Lung Cancer Compound Library | Anti-Blood Cancer Compound Library | Anti-Liver Cancer Compound Library | Anti-Colorectal Cancer Compound Library | Protein-protein Interaction Inhibitor Library | Membrane Protein-targeted Compound Library | Membrane Receptor-targeted Compound Library | Rulonilimab | PD-1/PD-L1-IN-19 | [D-Leu-4]-OB3 | NSC622608 | Sulindac | BMS-1166 | PD-1/PD-L1-IN-18 | Pacmilimab | Anti-Mouse PD-L1 Antibody | Vudalimab | PD-1/PD-L1-IN-24 | Cetrelimab | Human PD-L1 inhibitor III | PD-1/PD-L1-IN-20 | PD-1-IN-20 | PD-1/PD-L1-IN 5 | Sintilimab | PD-1/PD-L1-IN-9 hydrochloride | Nivolumab | PD-1/PD-L1-IN-16 | WL12 | PD-1/PD-L1-IN 6 | Acasunlimab | PD-1/PD-L1-IN-14 | PD1-PDL1-IN 1 | Sugemalimab | MAX-10181 | PD-1/PD-L1-IN-23 | D18
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Trending products:Recombinant Proteins | Bioactive Screening Libraries | Natural Products | Fluorescent Dye | PROTAC | Isotope-Labeled Compounds | Oligonucleotides | Antibodies | Click Chemistry
货号: HY-134886
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