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CAS No. :
MCE 国际站:GB-110 hydrochloride
产品活性:GB-110 hydrochloride 是一种有效的,具有口服活性的,非肽类的 protease activated receptor 2 (PAR2) 激动剂。GB-110 hydrochloride 选择性诱导 PAR2 介导的 HT29 细胞内 Ca2+ 释放,EC50 值为 0.28 μM。
研究领域:GPCR/G Protein
作用靶点:Protease Activated Receptor (PAR)
In Vitro: In an intracellular Ca2+ (iCa2+) mobilization assay using HT29 colon cancer cells, GB110 (EC50 240±20 nM; pEC50 6.7±0.05) is equipotent with the peptide agonist 2f-LIGRLO-NH2 (EC50 210±30 nM; pEC50 6.6±0.05), 10-fold more potent than SLIGRL-NH2, but ~35-fold less potent than trypsin (EC50 6±0.5 nM; pEC50 8.2±0.8).
相关产品:Bioactive Compound Library Plus | GPCR/G Protein Compound Library | Immunology/Inflammation Compound Library | Anti-Cancer Compound Library | Orally Active Compound Library | Targeted Diversity Library | Coagulation and Anti-coagulation Compound Library | Heterocyclic Compound Library | Membrane Protein-targeted Compound Library | Membrane Receptor-targeted Compound Library | Highly Selective Activators Library | Protease-Activated Receptor-3 (PAR-3) (1-6), human | I-191 | FSLLRY-NH2 TFA | VKGILS-NH2 | AC-55541 | FR-171113 | Protease-Activated Receptor-1 antagonist 3 | PAR-4 Agonist Peptide, amide TFA | Aeruginosin 98-B | AZ3451 | 2-Furoyl-LIGRLO-amide | AC-264613 | tcY-NH2 | ENMD-1068 hydrochloride | SLIGRL-NH2 | Protease-Activated Receptor-1, PAR-1 Agonist | CBK289001 | PAR-4 Agonist Peptide, amide | GB-88 | RWJ-56110 | Trypsin (MS grade) | AZ8838 | TRAP-6 | UDM-001651 | Parmodulin 2 | TFLLR-NH2 | Vorapaxar | SCH79797 dihydrochloride | TRAP-6-IN-1
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