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Prasugrel

CAS No. : 150322-43-3

MCE 国际站：Prasugrel

产品活性：Prasugrel，一种噻吩吡啶和前体，抑制血小板功能。Prasugrel 是一种具有口服活性的，有效的 P2Y12 受体拮抗剂，抑制 ADP 诱导的血小板聚集。

研究领域：GPCR/G Protein

作用靶点：P2Y Receptor

In Vivo: In rat platelets, Prasugrel active metabolite inhibits in vitro platelet aggregation induced by adenosine ADP (10μM) with an IC₅₀ value of 1.8 μM.
Prasugrel acts faster and is significantly more potent than Clopidogrel in vivo. Prasugrel is an inactive prodrug that requires metabolic processing in vivo to generate the active antiplatelet metabolite. Prasugrel is rapidly absorbed from the gut. After oral administration of standard-loading doses of 60 mg, maximum plasma levels of the active metabolite are achieved within 1 h, effective, maximum inhibition of platelet aggregation at 1-2 h.

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