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Urapidil

CAS No. : 34661-75-1

MCE 国际站：Urapidil

产品活性：Urapidil 是 α1 肾上腺素受体的拮抗剂和 5-HT_1A 受体的激动剂。

研究领域：GPCR/G Protein  |  Neuronal Signaling

作用靶点：5-HT Receptor  |  Adrenergic Receptor

In Vitro: Urapidil is an α1 adrenoreceptor antagonist and a 5-HT_1A receptor agonist. Urapidil does not affect vascular tone at concentrations up to 10^-5 M. Urapidil (10^-5 M) markedly inhibits the alpha 1-adrenergic agonist (phenylephrine)-induced concentration-dependent contractions in aortic rings without endothelium and also to some extent in those with endothelium. Moreover, the inhibitory effect of Urapidil is more pronounced in rings without endothelium than in those with endothelium. Urapidil (10^-5 M) affects neither the vascular tone nor the concentration-dependent contraction to serotonin.

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