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CAS No. : 81382-51-6
MCE 国际站:Pentiapine
产品活性:Pentiapine (CGS 10746) 是一种多巴胺释放 (dopamine release) 抑制剂,不与突触多巴胺受体位点结合。
研究领域:GPCR/G Protein | Neuronal Signaling
作用靶点:Dopamine Receptor
In Vivo: Pentiapine is a novel dopamine release inhibitor.The results show that Pentiapine dose-dependently reduces motor activity of mice. Moreover, Pentiapine dose-dependently reduces morphine-induced hyperactivity. Newman-Keuls post-hoc comparisons indicate that the group receiving morphine plus saline presents more activity than the groups receiving morphine plus 2 (P<0.05), 4, 8, 16, 24 and 32 (P<0.01) mg/kg of Pentiapine. Moreover, the groups receiving morphine plus 0.5, 1 and 2 mg/kg of Pentiapine present more activity than the groups receiving morphine plus 4, 8, 16, 24 and 32 mg/kg of Pentiapine (P<0.01). 30 mg/kg dose of Pentiapine completely blocks the methylenedioxymethamphetamine (MDMA) conditioned place preference (CPP) and also blocks the establishment of a cocaine CPP.
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货号: HY-100143
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