MCE 的所有产品仅用作科学研究或药证申报,我们不为任何个人用途提供产品和服务。
CAS No. : 635-12-1
MCE 国际站:1,4-Anthraquinone
产品活性:1,4-Anthraquinone 是一种有效的抗癌剂。1,4-Anthraquinone 阻断核苷转运,抑制大分子合成,诱导 DNA 碎片化,降低癌细胞生长和活力。1,4-Anthraquinone 可用于抗白血病研究。
研究领域:Cell Cycle/DNA Damage
作用靶点:DNA/RNA Synthesis
In Vitro: 1,4-Anthraquinone (2.62 nM-1.6 μM; 4 days) induces significant antiproliferative and cytotoxic effects in L1210 cells after 4 days at 6.55 nM; inhibits cell viability with IC50s of 100 nM at day 2 and 25 nM at day 4.
1,4-Anthraquinone (40.96 nM-25 μM; 30 min; L1210 cells) inhibits nucleoside transport by 71 and 92% and DNA synthesis by 84 and 96% at 4 and 10 μM, respectively, and are both irreversible upon drug removal.
1,4-Anthraquinone (0.1024-25 μM; 3 h) inhibits the rates of RNA and protein syntheses (IC50 = 2 μM) in a dose-dependent manner.
相关产品:Natural Product-like Compound Library | Bioactive Compound Library Plus | Cell Cycle/DNA Damage Compound Library | Anti-Cancer Compound Library | Fragment Library | Anti-Aging Compound Library | Anti-Blood Cancer Compound Library | IBU-DC Phosphoramidite | 2,4-D sodium salt | N6-Benzoyl-2'-deoxy-5'-O-DMT-a-adenosine 3'-CE phosphoramidite | Thailanstatin D | Carboplatin-d4 | Caracemide | N-DMTr-Morpholino-U-5'-O-phosphoramidite | Farudodstat | Ara-ATP | DNA31 | 2'-OMe-Ac-C Phosphoramidite | hDHODH-IN-12 | Dasabuvir | DNA Gyrase-IN-4 | Uridine triphosphate-13C9,15N2 sodium | 5-Methylcytosine | Cidofovir dihydrate | Capecitabine-d11 | DMT-2'-F-dA(bz) phosphoramidite | Tezacitabine | Mequindox | 5-Methylcytosine-d4 | TH287 hydrochloride | DNA Gyrase-IN-1 | DMT-2'-F-Cytidine Phosphoramidite | 2'-O-MOE-5-Me-rU | Levofloxacin sodium | GC7 Sulfate | Psammaplin A | hDHODH-IN-2
热门产品线:重组蛋白 | 化合物库 | 天然产物 | 荧光染料 | PROTAC | 同位素标记物 | 寡核苷酸 | 抗体 | 点击化学
Trending products:Recombinant Proteins | Bioactive Screening Libraries | Natural Products | Fluorescent Dye | PROTAC | Isotope-Labeled Compounds | Oligonucleotides | Antibodies | Click Chemistry
品牌介绍:
• MCE (MedChemExpress) 拥有200 多种全球独家化合物库,我们致力于为全球科研客户提供前沿最全的高品质小分子活性化合物;
• 50,000 多种高选择性抑制剂、激动剂涉及各热门信号通路及疾病领;
• 产品种类涵盖各种重组蛋白,多肽,常用试剂盒 ,更有 PROTAC、ADC 等特色产品,广泛应用于新药研发、生命科学等科研项目;
• 提供虚拟筛选,离子通道筛选,代谢组学分析检测分析,药物筛选等专业技术服务;
• 设有专业的实验中心和严格的质控、验证体系;
• 提供 LC/MS、NMR、HPLC、手性分析、元素分析等各项质检报告,确保产品的高纯度、高品质;
• 产品的生物活性多经各国客户实验验证;
• Nature, Cell, Science 等多种顶级期刊及制药专利收录了MCE客户的科研成果;
• 专业团队跟踪最新的制药及生命科学研究进展,为您提供全球最新的活性化合物;
• 与世界各大制药公司及知名科研机构建立了长期的合作。