MCE 的所有产品仅用作科学研究或药证申报,我们不为任何个人用途提供产品和服务。
SB 243213 dihydrochloride
CAS No. : 1780372-25-9
MCE 国际站:SB 243213 dihydrochloride
产品活性:SB 243213 dihydrochloride 是一种口服有效的,选择性的,高亲和力的 5-HT2C 受体拮抗剂,对人 5-HT2C 受体的 pKi 为 9.37,pKb 为 9.8。SB 243213 dihydrochloride 对多种神经递质受体、酶和离子通道具有超过 100 倍的选择性。SB 243213 dihydrochloride 具有改善的抗焦虑特性,有用于精神分裂症和运动障碍的潜力。
研究领域:GPCR/G Protein | Neuronal Signaling
作用靶点:5-HT Receptor
In Vitro: SB 243213 dihydrochloride shows little affinity (pKi<6) for cloned human 5-HT1A, 5-HT1B, 5-HT1E, 5- HT1F and 5-HT7 receptors. It shows weak affinity (pKi<6.5) for the cloned human 5-HT1D and D3 receptors and moderate affinity (pKi=6.7) for the cloned human D2 receptor.
SB 243213 dihydrochloride shows 100-fold selectivity over a wide range of neurotransmitter receptors, enzymes and ion channels.
In Vivo: SB 243213 dihydrochloride (0.1-10 mg/kg; p.o.; 1 h pre-test) dose-dependently and significantly increases the amount of time rats spent in social interaction over 15 min under brightly lit conditions and in an unfamiliar test box.
SB 243213 dihydrochloride (0.3 mg/kg; p.o.; 1 h pre-test) significantly increases time spent in social interaction.
相关产品:Chlorpromazine hydrochloride | Serotonin hydrochloride | SCH-23390 hydrochloride | Harmine | Puerarin | PNU-282987 | Clozapine | Scopolamine hydrobromide | Risperidone | Dihydroergotamine mesylate | Olanzapine | GTS-21 dihydrochloride | Vortioxetine | Aripiprazole | Amitriptyline hydrochloride | Ondansetron | Thioridazine hydrochloride | Brexpiprazole | SB-269970 hydrochloride | SEP-363856 hydrochloride | Cisapride | Volinanserin | 8-OH-DPAT | Ketanserin | Pimavanserin | Pindolol
热门产品线:重组蛋白 | 药物筛选 | 天然产物 | 荧光染料 | PROTAC | 同位素标记物
Trending products:Recombinant Proteins | Bioactive Screening Libraries | Natural Products | Dye Reagents | PROTAC | Isotope-Labeled Compounds
品牌介绍:
• MCE (MedChemExpress) 拥有200 多种全球独家化合物库,我们致力于为全球科研客户提供前沿最全的高品质小分子活性化合物;
• 50,000 多种高选择性抑制剂、激动剂涉及各热门信号通路及疾病领域;
• 产品种类涵盖各种重组蛋白,多肽,常用试剂盒 ,更有 PROTAC、ADC 等特色产品,广泛应用于新药研发、生命科学等科研项目;
• 提供虚拟筛选,离子通道筛选,代谢组学分析检测分析,药物筛选等专业技术服务;
• 设有专业的实验中心和严格的质控、验证体系;
• 提供 LC/MS、NMR、HPLC、手性分析、元素分析等各项质检报告,确保产品的高纯度、高品质;
• 产品的生物活性多经各国客户实验验证;
• Nature, Cell, Science 等多种顶级期刊及制药专利收录了MCE客户的科研成果;
• 专业团队跟踪最新的制药及生命科学研究进展,为您提供全球最新的活性化合物;
• 与世界各大制药公司及知名科研机构建立了长期的合作。