耗材描述
Urabrelimab
产品活性:Urabrelimab (SRF231) 是一种完全人抗 CD47 单克隆抗体,可阻断 CD47-SIRP 相互作用。
产品来源: https://www.medchemexpress.cn/urabrelimab.html
研究领域:Immunology/Inflammation
作用靶点:Interleukin Related
In Vitro: Urabrelimab (SRF231) promotes macrophage-mediated phagocytic clearance of several hematologic primary tumor samples and cell lines in vitro. Urabrelimab increases phagocytosis of Raji tumor cell line targets with an EC50 of ~300 ng/mL.
In Vivo: Urabrelimab (SRF231) administration leads to profound tumor growth inhibition in models of multiple myeloma, diffuse large B cell lymphoma and Burkitt's lymphoma as a single agent and in combination with opsonizing antibodies. In the Raji xenograft model, single agent therapy leads to 112% tumor growth inhibition.
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