耗材描述
Men 10376 TFA
产品活性:Men 10376 TFA 是一种有效的选择性的 tachykinin NK-2 受体拮抗剂,对大鼠小肠 NK-2 受体的 Ki 值为 4.4 μM。
产品来源: https://www.medchemexpress.cn/Men_10376_TFA.html
研究领域:GPCR/G Protein | Neuronal Signaling
作用靶点:Neurokinin Receptor
In Vitro: Men 10376 is a selective tachykinin NK-2 receptor, with a Ki of 4.4 μM, and shows low selectivity for NK-1 and NK-3 receptors (Ki, >10 μM). Men 10376 shows pA2s of 5.66 and 8.08 for NK-1 (guinea-pig ileum) and NK-2 receptors (endothelium-deprived rabbit pulmonary artery). Men 10376 shows no effect on NK-3 receptor (Ki, >10 μM).
In Vivo: Men 10376 (1 and 3 μmol/kg) antagonizes increase in bladder motility produced by the NK-2 receptor agonist in rats.
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