耗材描述
Magainin 1 TFA
产品活性:Magainin 1 TFA (Magainin I TFA) 是从 Xenopus laevis 皮肤中分离出的一种抗菌和两亲性肽。Magainin 1 TFA 对多种革兰氏阴性和革兰氏阳性细菌均表现出抗生素活性。
产品来源: https://www.medchemexpress.cn/magainin-1-tfa.html
研究领域:Anti-infection
作用靶点:Bacterial | Fungal | Antibiotic
结构分类:其他类 | 结构分类
In Vitro: Magainin 1 interacts with acidic lipids through electrostatic interactions followed by hydrophobic interactions to form an amphiphilic helix, inducing the leakage. Magainin 1 induces the leakage of calcein specifically out of negatively-charged vesicles. The peptide binds to bovine brain phosphatidylserine sonicated vesicles according to the Langmuir isotherm with a binding constant of 3.8×105 M-1 and a binding-site number of 0.10 per lipid molecule.
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