耗材描述
Porcine dynorphin A(1-13)
产品活性:Porcine dynorphin A (1-13) 是一个有效的内源性阿片受体 (κ opioid receptor) 激动剂,在生理浓度下它有缓解疼痛作用。
产品来源: https://www.medchemexpress.cn/Porcine-dynorphin-A_1-13_.html
研究领域:GPCR/G Protein | Neuronal Signaling
作用靶点:Opioid Receptor
In Vivo: Dynorphin A (1-13) exposure (33 μM) causes a significant loss in neuronal viability at 4 h with a visible destruction in neuronal morphology seen at 16 h. Exposure to dynorphin A (1-13) causes acute increases in [Ca2+]i in individual neurons similar to increases seen with acute NMDA treatment. Continuous exposure to dynorphin A (1-13) (100 μM) causes a significant loss of neurons over time.
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