耗材描述
Contulakin G
产品活性:Contulakin G 是一种 O-糖基化无脊椎动物神经紧张素。Contulakin-G 是一种较弱的神经紧张素受体 (neurotensin receptor) 激动剂。Contulakin G 还是一种有效的镇痛剂。
产品来源: https://www.medchemexpress.cn/contulakin-g.html
研究领域:GPCR/G Protein | Neuronal Signaling
作用靶点:Neurotensin Receptor
In Vivo: Contulakin G exhibits potent analgesic activity in three pain models in rats following intrathecal delivery, namely in tail-flick (acute pain), formalin test, and CFA-induced allodynia inflammatory pain.
Contulakin G (0-3 nmoL, Intrathecally) significantly decreases flinching behavior in rats.
Contulakin G (50-500 nmoL, Intrathecally) produces a dose-dependent increase in the thermally evoked skin twitch latency by 30 min after administration in dogs.
相关产品:AF38469 | Neurotensin | SBI-553 | LM11A-31 dihydrochloride | Neurotensin(8-13) | THX-B | SORT-PGRN interaction inhibitor 1 | AF40431 | SR 142948 dihydrochloride | ML314 | Latozinemab | Kinetensin | [Lys8, Lys9]-Neurotensin (8-13) | Levocabastine hydrochloride | Sortilin antagonist 1 | JMV 449 acetate | NTRC-824 | (S)-Osanetant | Acetyl neurotensin (8-13) | BVFP | hNTS1R agonist-1 | SORT-PGRN interaction inhibitor 3 | VGD071 | [D-Trp11]-Neurotensin
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