耗材描述
Myriocin
产品活性:Myriocin (Thermozymocidin) 是一种可以从 Myriococcum albomyces, Isaria sinclairi 和 Mycelia sterilia 中分离的真菌代谢产物,是一种有效的丝氨酸-棕榈酰转移酶 (SPT) 抑制剂,是鞘脂从头合成的关键。Myriocin 抑制亚基因组 HCV-1b 复制子和基因型 2a 感染性 HCV 的 JFH-1 株的复制,抑制 HCV 感染的 IC50 为 3.5 μg/mL。
产品来源: https://www.medchemexpress.cn/myriocin.html
研究领域:Anti-infection
作用靶点:HCV | Antibiotic
结构分类:酮、醛、酸 | 结构分类
In Vitro: Myriocin (Thermozymocidin; 0-10000 nM; 96 h; Huh7/Rep-Feo cells) inhibits the replication of a subgenomic hepatitis C virus (HCV) genotype 1b replicon.
Myriocin (100 nM; 72 h) decreases in the sphingomyelin content of Huh7 cells.
In Vivo: Myriocin (Thermozymocidin; 0-1 mg/kg; i.p.; daily, for 5 d; male Balb/c mice) blocks de novo synthesis of sphingolipids in vivo by SPT inhibition and induced c-myc expression in liver.
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