耗材描述
Rubropunctamine
产品活性:Rubropunctamine 是一种红色红曲色素。Rubropunctamine 不仅对细菌有抗菌作用,而且对某些酵母菌和丝状真菌菌株也有抗菌作用。Rubropunctamine 还具有潜在的胚胎毒性和致畸性。
产品来源: https://www.medchemexpress.cn/rubropunctamine.html
研究领域:Anti-infection
作用靶点:EBV | Fungal | Bacterial
结构分类:生物碱 | 异喹啉类生物碱 | 结构分类
In Vitro: Rubropunctamine (0.32-32 nM; 48 h) inhibits Epstein-Barr virus early antigen (EBV-EA) activation induced by 12-O-tetradecanoylphorbol-13-acetate (TPA), with an IC50 of 433 mol ratio/32 pmol TPA.
Rubropunctamine (1 h) exhibits moderate scavenging activity (inhibitory ratio (IR)=1.5) against NO generation by (±)-(E)-methyl-2[(E)-hydroxy-imino]-5-nitro-6-methoxy-3-hexemide (NOR 1) in normal human hepato cells.
In Vivo: Rubropunctamine inhibits TPA-induced inflammation in mice, with an ID50 of 0.32 mg/ear.
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