耗材描述
Clemastanin B
产品活性:Clemastanin B 是一种木质素,通过抑制病毒增殖、预防和阻断病毒附着而具有强大的抗流感 (anti-influenza) 活性。Clemastanin B 靶向病毒内吞作用、脱壳或核糖核蛋白 (RNP) 从细胞核输出。Clemastanin B 具有抗氧化和抗炎活性。
产品来源: https://www.medchemexpress.cn/clemastanin-b.html
研究领域:Anti-infection
作用靶点:Influenza Virus
来源:植物 | 十字花 | 板蓝根
结构分类:苯丙素类 | 木脂素
In Vitro: Clemastanin B inhibits different subtypes of human (H1N1, including swine-origin H1N1; H3N2 and influenza B) and avian influenza viruses (H6N2, H7N3, H9N2) at different magnitudes of activity (IC50 0.087-0.72 mg/ml) while this compound was inactive against respiratory syncytial virus (RSV), adenovirus 3 (ADV3), parainfluenza virus 3 (PIV3), enterovirus 71 (EV71) and human rhinovirus (HRV).
Clemastanin B (0.05, 0.1, 0.2, 0.4 mg/ml; for 8 hours) treatment results in nucleoprotein (NP) distribution in the nuclei in MDCK cells.
Clemastanin B (48-72 h) after virus incubation (MOI, 0.01; for 2 h) causes a pronounced titer reduction of progeny virus in MDCK cells.
Clemastanin B (pre-incubated for 2 h) has no protective effect on MDCK cell lines with influenza virus.
相关产品:Natural Product Library Plus | Bioactive Compound Library Plus | Anti-Infection Compound Library | Immunology/Inflammation Compound Library | Natural Product Library | Antiviral Compound Library | Antioxidant Compound Library | Glycoside Compound Library | Traditional Chinese Medicine Active Compound Library | Antiviral Traditional Chinese Medicine Active Compound Library | Anti-inflammatory Traditional Chinese Medicine Active Compound Library | Plant-Sourced Natural Product Library | Heterocyclic Compound Library | Radioprotector Library | Bioactive Compound Library Max | Acetylcysteine | Tunicamycin | Curcumin | U0126-EtOH | Camptothecin | Vadimezan | Indomethacin | Aprotinin | Rifampicin | Molnupiravir | Baicalein | Oseltamivir acid | Spermine | Geldanamycin | AEBSF hydrochloride | α-Vitamin E | Favipiravir | HA Peptide | Chlorogenic acid | 6-Diazo-5-oxo-L-nor-Leucine | Baloxavir | Tofacitinib citrate | Trimethoprim | AG-1478 | Harringtonine | YM-201636 | Isoliquiritigenin | SC75741
品牌介绍: MCE (MedChemExpress) 拥有数百种全球独家化合物,我们致力于为全球科研客户提供最新最全的高品质小分子活性化合物;10,000 多种高选择性抑制剂、激动剂涉及各热门信号通路及疾病领域;设有专业的实验中心和严格的质控、验证体系;提供 LC/MS、NMR、HPLC、手性分析、元素分析等各项质检报告,确保产品的高纯度、高品质;产品的生物活性多经各国客户实验验证;Nature, Cell, Science 等多种顶级期刊及制药专利收录了MCE客户的科研成果;专业团队跟踪最新的制药及生命科学研究进展,为您提供全球最新的活性化合物;与世界各大制药公司及知名科研机构建立了长期的合作。