耗材描述
Rebeccamycin
产品活性:Rebeccamycin,一种抗肿瘤抗生素,抑制 DNA 拓扑异构酶 I (DNA topoisomerase I)。Rebeccamycin 通过毒害拓扑异构酶 I 发挥其主要的抗肿瘤作用,对蛋白激酶 C 和拓扑异构酶 Ⅱ 的作用较小。
产品来源: https://www.medchemexpress.cn/rebeccamycin.html
研究领域:Cell Cycle/DNA Damage | Antibody-drug Conjugate/ADC Related | Anti-infection
作用靶点:Topoisomerase | ADC Cytotoxin | Antibiotic
结构分类:抗生素 | 疾病研究 | 抗癌 | 抗生素 | 其他类 | 结构分类
In Vitro: Rebeccamycin is an antitumor antibiotic produced by the actinomycete Saccharotrix aerocolonigenes with activity against several human tumor cell lines, including A549 (lung adenocarcinoma), HCT-116 (colon carcinoma), and KB (nasopharyngeal carcinoma) .
Rebeccamycin shows antibacterial activity against several Gram-positive bacteria, including Staphylococcus aureus and Streptococcus faecalis.
In Vivo: Rebeccamycin (2-256 mg/kg; i.p.; daily for 9 days) prolongs survival in B16 melanoma, L1210 leukemia.
相关产品:Rapamycin | Cycloheximide | Chloroquine | Doxorubicin hydrochloride | Bafilomycin A1 | Paclitaxel | Dexamethasone | Puromycin dihydrochloride | Staurosporine | Actinomycin D | Etoposide | G-418 disulfate | Monomethyl auristatin E | Nigericin sodium salt | Cyclosporin A | 5-Azacytidine | Brefeldin A | Bleomycin sulfate | Exatecan mesylate | Ionomycin | Hygromycin B | Mitomycin C | Resveratrol | Tunicamycin | Doxycycline hyclate | Tacrolimus | SN-38
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