耗材描述
ε-Amanitin
产品活性:ε-Amanitin,从多种蘑菇中分离出的环状肽,可有效与 RNA 聚合酶 II (RNA polymerase II) 结合并抑制其活性。
产品来源: https://www.medchemexpress.cn/ε-amanitin.html
研究领域:Cell Cycle/DNA Damage | Antibody-drug Conjugate/ADC Related
作用靶点:DNA/RNA Synthesis | ADC Cytotoxin
结构分类:酚类 | 单酚类 | 其他类
In Vitro: Amatoxin Family includes alpha-Amanitin, beta-Amanitin, gamma-Amanitin, epsilon-Amanitin (ε-Amanitin), Amanullin, Amanullinic acid, Amaninamide, Amanin and Proamanullin. Amatoxins are potent and selective inhibitors of RNA polymerase II, a vital enzyme in the synthesis of messenger RNA (mRNA), microRNA, and small nuclear RNA (snRNA). By inhibiting the synthesis of mRNA, Amatoxins thereby stop cell metabolism by inhibiting transcription and protein biosynthesis, which results in cellular apoptosis. Consequently Amatoxins stop cell growth and proliferation.
相关产品:Cycloheximide | Doxorubicin hydrochloride | Paclitaxel | Dexamethasone | Actinomycin D | Oxaliplatin | Gemcitabine | Monomethyl auristatin E | Bleomycin sulfate | Exatecan mesylate | Carboplatin | Mitomycin C | Cytarabine | 5-BrdU | SN-38 | Methotrexate | Streptozotocin | Camptothecin | Anisomycin | Fludarabine | ART558 | Propidium Iodide | Thymidine | Hydroxyurea | Mertansine | Daunorubicin hydrochloride | Remdesivir
品牌介绍: MCE (MedChemExpress) 拥有数百种全球独家化合物,我们致力于为全球科研客户提供最新最全的高品质小分子活性化合物;10,000 多种高选择性抑制剂、激动剂涉及各热门信号通路及疾病领域;设有专业的实验中心和严格的质控、验证体系;提供 LC/MS、NMR、HPLC、手性分析、元素分析等各项质检报告,确保产品的高纯度、高品质;产品的生物活性多经各国客户实验验证;Nature, Cell, Science 等多种顶级期刊及制药专利收录了MCE客户的科研成果;专业团队跟踪最新的制药及生命科学研究进展,为您提供全球最新的活性化合物;与世界各大制药公司及知名科研机构建立了长期的合作。