耗材描述
OMDM-1
产品活性:OMDM-1 是一种有效选择性的,代谢稳定的 anandamide 细胞摄取 (ACU) 抑制剂,Ki 值为2.4 μM。
产品来源: https://www.medchemexpress.cn/omdm-1.html
研究领域:Metabolic Enzyme/Protease
作用靶点:Endogenous Metabolite
结构分类:生物碱 | 其他类生物碱 | 酚类 | 单酚类 | 结构分类
In Vitro: OMDM-1 shows poor affinity for either CB1 (Ki=12.1 μM) or CB2 (Ki>10 μM) receptors in rat brain and spleen membranes, respectively; OMDM-1 has almost no activity at vanilloid receptors in the intracellular calcium assay carried out with intact cells over-expressing the human VR1 (EC50≥10 μM), and no activity as inhibitors of FAAH in N18TG2 cell membranes (Ki>50 μM).
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