耗材描述
Licopyranocoumarin
产品活性:Licopyranocoumarin 是一种异黄酮,具有 CYP3A4 抑制活性,IC50 为 32 μM。Licopyranocoumarin 具有有效的神经保护活性。
产品来源: https://www.medchemexpress.cn/licopyranocoumarin.html
研究领域:Metabolic Enzyme/Protease
作用靶点:Cytochrome P450
来源:植物 | 豆科 | 甘草
结构分类:苯丙素类 | 香豆素 | 结构分类
In Vitro: Licopyranocoumarin (0.3-3 μM; 48 hours) markedly blocks MPP+-induced neuronal PC12D cell death and disappearance of mitochondrial membrane potential, which were mediated by JNK.
Licopyranocoumarin (0.3-3 μM; 36 hours) inhibits MPP+-induced JNK activation through the suppression of reactive oxygen species (ROS) generation, thereby inhibiting MPP+-induced neuronal PC12D cell death.
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