耗材描述
AC-VEID-CHO TFA
产品活性:AC-VEID-CHO (TFA) 是一种多肽来源的半胱天冬酶抑制剂,对 Caspase-6、Caspase-3 和 Caspase-7 具有抑制作用,IC50 值分别为 16.2 nM、13.6 nM 和162.1 nM。AC-VEID-CHO (TFA) 可被用于阿尔茨海默病、亨廷顿病等神经退行性疾病的研究。
产品来源: https://www.medchemexpress.cn/ac-veid-cho-tfa.html
研究领域:Apoptosis
作用靶点:Caspase
In Vitro: AC-VEID-CHO (TFA) has potency of inhibition for Caspase-6, Caspase-3 and Caspase-7 with IC50 values of 16.2 nM, 13.6 nM and 162.1 nM, respectively.
Ac-VEID-CHO is predominantly excluded from accessing the intracellular environment (0.16% cellular accumulation) and lacks any activity with an IC50 value of >100 μM in the cellular assay.
AC-VEID-CHO (TFA) (also inactive in lamin degradation assay) is clearly able to inhibit VEIDase activity with an IC50 value of 0.49 μM when the membrane barrier is removed.
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