耗材描述
Adenosine N1-oxide
产品活性:Adenosine N1-oxide 是一种具有口服活性的抗炎剂,可从蜂王浆中分离得到。Adenosine N1-oxide 促进成骨和成脂分化。
产品来源: https://www.medchemexpress.cn/adenosine-n1-oxide.html
研究领域:Others
作用靶点:Others
结构分类:其他类 | 结构分类
In Vitro: Adenosine N1-oxide )(1-40 μM, 24 h) inhibits TNF-α and IL-6 secretion by RAW264.7 cells stimulated with 2 µg/mL LPS (HY-D1056).
Adenosine N1-oxide )(20/100 μM, 30 mins) increases intracellular cAMP production in both peritoneal macrophages and RAW264.7 cells in a dose-dependent manner.
Adenosine N1-oxide )(5-10 μM, 30 mins) increases the protein level of phosphorylation of Akt and GSK-3β in 2 µg/mL LPS (HY-D1056)-stimulated RAW264.7 cells.
Adenosine N1-oxide )(2-10 μM, 6-7 days) promotes osteogenic and adipocyte differentiation in MC3T3-E1 cells.
In Vivo: Adenosine N1-oxide (oral administration, 135 mg/kg for three times) reduces the lethality caused by LPS (HY-D1056)-induced endotoxin shock in BALB/c mice.
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