耗材描述
Ropinirole-d7 hydrochloride
产品活性:Ropinirole-d7 (hydrochloride) 是 Ropinirole hydrochloride 的氘代物。 Ropinirole (SKF 101468) hydrochloride 是一种口服有效的 D3/D2 受体激动剂,对 D2 受体的 Ki 为 29 nM。Ropinirole hydrochloride 对 hD2,hD3 和 hD4 受体的 pEC50 分别为 7.4、8.4 和 6.8。Ropinirole hydrochloride 对 D1 受体没有亲和力。Ropinirole hydrochloride 具有用于帕金森氏病潜力。
产品来源: https://www.medchemexpress.cn/ropinirole-d7-hydrochloride.html
研究领域:GPCR/G Protein | Neuronal Signaling
作用靶点:Dopamine Receptor
In Vitro: Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs.
相关产品:Clozapine N-oxide | MPTP hydrochloride | Oxidopamine hydrobromide | Chlorpromazine hydrochloride | L-DOPA | Dopamine hydrochloride | SCH-23390 hydrochloride | Haloperidol | Pimozide | SKF 38393 hydrochloride | Risperidone | Cabergoline | Olanzapine | Aripiprazole | Bromocriptine mesylate | Fluphenazine dihydrochloride | ONC206 | Thioridazine hydrochloride | Brexpiprazole | Sulpiride | Trifluoperazine dihydrochloride | Flunarizine dihydrochloride | Quinpirole hydrochloride | WAY-100635 maleate | Quetiapine | Lurasidone
品牌介绍: MCE (MedChemExpress) 拥有数百种全球独家化合物,我们致力于为全球科研客户提供最新最全的高品质小分子活性化合物;10,000 多种高选择性抑制剂、激动剂涉及各热门信号通路及疾病领域;设有专业的实验中心和严格的质控、验证体系;提供 LC/MS、NMR、HPLC、手性分析、元素分析等各项质检报告,确保产品的高纯度、高品质;产品的生物活性多经各国客户实验验证;Nature, Cell, Science 等多种顶级期刊及制药专利收录了MCE客户的科研成果;专业团队跟踪最新的制药及生命科学研究进展,为您提供全球最新的活性化合物;与世界各大制药公司及知名科研机构建立了长期的合作。