耗材描述
Glipizide-d11
产品活性:Glipizide-d11 是 Glipizide 的氘代物。Glipizide (CP 2872; K 4024) 是一种有效的、具有口服活性的磺酰脲类抗糖尿病试剂 (anti-diabetic agent),可用于 2 型糖尿病的研究,但不适用于1 型糖尿病。Glipizide 通过部分阻断郎格汉斯胰岛细胞中 ATP 敏感钾通道 (KATP) 发挥作用。
产品来源: https://www.medchemexpress.cn/glipizide-d11.html
研究领域:Membrane Transporter/Ion Channel
作用靶点:Potassium Channel
In Vitro: Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs.
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