耗材描述
SBC-115076
产品活性:SBC-115076 是一种有效的前蛋白转化酶枯草杆菌蛋白酶/ kexin 9型 (PCSK9) 抑制剂。PCSK9 是一种前蛋白转化酶,在 LDL 受体代谢中起重要作用。
产品来源: https://www.medchemexpress.cn/SBC-115076.html
研究领域:Metabolic Enzyme/Protease
作用靶点:Ser/Thr Protease
In Vivo: SBC-115076 (4 mg/kg; s.c.; daily for 3 weeks) reduces obesity and dyslipidemia, as well as improves insulin sensitivity in HFD-fed rats.
相关产品:Bioactive Compound Library Plus | Metabolism/Protease Compound Library | Peptidomimetic Library | Anti-Cardiovascular Disease Compound Library | Lipid Metabolism Compound Library | Targeted Diversity Library | Coagulation and Anti-coagulation Compound Library | Heterocyclic Compound Library | Protease Inhibitor Library | Bioactive Compound Library Max | Leupeptin hemisulfate | Aprotinin | AEBSF hydrochloride | Proteinase K | Camostat mesylate | WNK463 | Bradykinin | Nafamostat mesylate | Trypsin | Inclisiran | Trypsin Inhibitor, soybean | Evolocumab | Benzamidine hydrochloride | PF-06446846 hydrochloride | Chymotrypsin | WNK-IN-11 | Bococizumab | Pep2-8 | Avoralstat | IPR-803 | Alirocumab | Inclisiran sodium | Berotralstat dihydrochloride | TPCK | UK122 | UKI-1 | Sebetralstat | PCSK9-IN-12 | R-IMPP | BioE-1115
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