耗材描述
PDGFRα kinase inhibitor 1
产品活性:PDGFRα kinase inhibitor 1 是一种高选择性 II 型 PDGFRα 激酶抑制剂,抑制 PDGFRα 和 PDGFRβ 的 IC50 分别为 132 nM 和 6115 nM。
产品来源: https://www.medchemexpress.cn/PDGFR_alpha__kinase_inhibitor_1.html
研究领域:Protein Tyrosine Kinase/RTK
作用靶点:PDGFR
In Vitro: PDGFRα kinase inhibitor 1 (CHMFL-PDGFR-159, Compound 15i) exhibits weak inhibition to DDR1 kinase (IC50: 2462±126 nM).
相关产品:Bioactive Compound Library Plus | Kinase Inhibitor Library | Protein Tyrosine Kinase Compound Library | Anti-Cancer Compound Library | Reprogramming Compound Library | Angiogenesis-Related Compound Library | Targeted Diversity Library | Anti-Liver Cancer Compound Library | Anti-Pulmonary Fibrosis Compound Library | Membrane Protein-targeted Compound Library | Membrane Receptor-targeted Compound Library | Highly Selective Inhibitors Library | Cytokine Inhibitors Library | Multi-Target Compound Library | Bioactive Compound Library Max | Anti-Fibrosis Compound Library | Lenvatinib | Regorafenib | Sunitinib | Nintedanib | Imatinib | Ponatinib | Axitinib | Pazopanib | Crenolanib | SU 5402 | Avapritinib | Linifanib | CP-673451 | Ripretinib | Masitinib | Dovitinib | Cediranib | CHIR-124 | Tyrphostin A9 | Sennoside B | Narazaciclib | Amuvatinib
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