耗材描述
Otenzepad
产品活性:Otenzepad (AF-DX 116) 是一种选择性的、竞争性的 M2 毒蕈碱乙酰胆碱受体拮抗剂,对兔外周肺和大鼠心脏的 IC50 值分别为 640 nM 和 386 nM。
产品来源: https://www.medchemexpress.cn/otenzepad.html
研究领域:GPCR/G Protein | Neuronal Signaling
作用靶点:mAChR
In Vivo: Otenzepad (0.5, 1 mg/kg, s.c., in rats) significantly improved win-stay acquisition relative to vehicle-injected controls.
Otenzepad (2 mg/kg, s.c., in rats) significantly improved retention relative to vehicle controls.
Otenzepad (0.3, 1.0, or 3.0 mg/kg, ip, in mice) potentiates the effects of glucose and reverses the effects of insulin on memory.
相关产品:Drug Repurposing Compound Library Plus | Clinical Compound Library Plus | Bioactive Compound Library Plus | GPCR/G Protein Compound Library | Neuronal Signaling Compound Library | Clinical Compound Library | Drug Repurposing Compound Library | Neurotransmitter Receptor Compound Library | Anti-Parkinson's Disease Compound Library | Neurodegenerative Disease-related Compound Library | Heterocyclic Compound Library | Membrane Protein-targeted Compound Library | Membrane Receptor-targeted Compound Library | Highly Selective Inhibitors Library | Bioactive Compound Library Max | Clozapine N-oxide | Deschloroclozapine | Pilocarpine Hydrochloride | Atropine | Scopolamine hydrobromide | Carbamoylcholine chloride | Olanzapine | Amitriptyline hydrochloride | Methacholine chloride | Xanomeline | Mepenzolate bromide | (S)-(+)-Dimethindene maleate | Promethazine hydrochloride | Propantheline bromide | Benztropine mesylate | Oxotremorine M iodide | Arecoline hydrobromide | Darifenacin hydrobromide | Tiotropium Bromide | DREADD agonist 21 | Pirenzepine dihydrochloride | Dronedarone
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