耗材描述
Multi-kinase-IN-1
产品活性:Multi-kinase-IN-1 (Compound 11k) 是一种具有抗肿瘤活性的激酶 (kinase) 抑制剂。Multi-kinase-IN-1 诱导细胞凋亡 (apoptosis),可用于结直肠癌的研究。
产品来源: https://www.medchemexpress.cn/multi-kinase-in-1.html
研究领域:Apoptosis | Protein Tyrosine Kinase/RTK
作用靶点:Apoptosis | c-Met/HGFR | PDGFR | Src | TAM Receptor
In Vitro: Multi-kinase-IN-1 (Compound 11k) (0-5 µg/mL, 0-72 h) induces antiproliferation and cytotoxicity in a dose- and time-dependent manner in HT-29 cells, and is much less toxic to normal colorectal mucosa epithelial cells.
Multi-kinase-IN-1 (0-3 µg/mL, 0-72 h) induces cell apoptosis in a time- and dose-dependent manner.
Multi-kinase-IN-1 (0-3 µg/mL, 48 h) slightly induces cell cycle arrest in G2/M phase.
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