耗材描述
Antiparasitic agent-9
产品活性:Antiparasitic agent-9 (compound 47) 是一种口服有效的抗寄生虫剂。Antiparasitic agent-9 显示对人类寄生虫的抗寄生虫活性。
产品来源: https://www.medchemexpress.cn/antiparasitic-agent-9.html
研究领域:Anti-infection
作用靶点:Parasite
In Vivo: Antiparasitic agent-9 (compound 47) (15 mg/kg, Orally, twice each day for 7 days) reduces adult worm burden in the jird L. sigmodontis infection model.
Antiparasitic agent-9 (2 mg/kg (IV), 10 and 30 mg/kg (PO); once) shows a brain to plasma ratio of 0.08, suggesting limited brain exposure.
Pharmacokinetic Parameters of Antiparasitic agent-9 in male Male CD-1 mouse.
PO (30 mg/kg)
PO (10 mg/kg)
IV (2 mg/kg)
Cmax (μM)
13.9
5.27 ± 0.83
Tmax (h)
0.50
4.0 ± 2.8
AUC0-inf (μM·h)
121
68.1±NC
CL (mL/min/kg)
3.6 ± 0.22
Vd ss (mL/kg)
0.74 ± 0.08
F (%)
57
brain/plasma [b]/[p]
0.08
efflux ratio (ER)
12
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