Product Introduction
Bioactivity


英文名: EC5026

描述: EC5026 (BPN-19186) 是首创的，非阿片类的，可溶性环氧水解酶 (sEH) 抑制剂，它可有效缓解发炎性和神经性疼痛。

体内活性: EC5026（BPN-19186）是一类先锋小分子，它能强效抑制关键调节酶——可溶性环氧化合酶（sEH）。EC5026 抑制 sEH 可通过稳定天然镇痛和抗炎介质来治疗疼痛。EicOsis开发的sEH抑制剂在实验室动物中已显示出有效缓解疼痛，且没有明显的不良或成瘾性副作用，并且能缓解犬、猫及马自然发生的疼痛。

存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year

溶解度: DMSO : 250 mg/mL (616.69 mM)


关键字: sEH | analgesic | Epoxide Hydrolase | BPN 19186 | pain | inhibit | Hydrolase | anti-inflammatory | Inhibitor | EC5026 | mediators | Epoxide | EC 5026 | BPN19186 | EC-5026 | Soluble

相关产品: 1-Cyclohexyl-3-dodecyl urea | AUDA | beta-Amyrin acetate | trans-AUCB | Valpromide | PTUPB | (Rac)-EC5026 | N,N'-Dicyclohexylurea | BI-1935 | ARM1

相关库: Anti-Aging Compound Library | Bioactive Compounds Library Max | Inhibitor Library | Anti-Fibrosis Compound Library | Metabolism Compound Library | Preclinical Compound Library | Covalent Inhibitor Library | NO PAINS Compound Library | Bioactive Compound Library