Product IntroductionBioactivity英文名:
Arimoclomol citrate描述: Arimoclomol citrate (BRX-220 citrate) is a heat shock protein (HSP) co-inducer that acts by enhancing Hsp expression and directly impacting protein aggregation, clearance of misfolded assemblies, and the proteasome-ubiquitin system. This compound is known for its ability to protect motor neurons.
体内活性: Arimoclomol (BRX-220; 20 mg/kg; orally administered for 5 d) has a protective effect against cholecystokinin-octapeptide (CCK)-induced acute pancreatitis[1]. Animal Model: Male Wistar rats weighing 240 to 270 g[1]Dosage: 20 mg/kg Administration: Administered intragastrically, for 5 days Result: Had a protective effect against CCK-induced acute pancreatitis.
存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year
关键字:
BRX 220 Citrate |
BRX220 Citrate |
Arimoclomol Citrate |
BRX-220 Citrate