Product Introduction
Bioactivity


英文名: PBRM1-BD2-IN-8

描述: PBRM1-BD2-IN-8 (compound 34) 是一种强效的 PBRM1 Bromodomain 抑制剂 (PBRM1-BD2 Kd=4.4 μM, PBRM1-BD2 IC50=0.16 μM; PBRM1-BD5 Kd=25 μM)，其具有抗癌活性。

体外活性: PBRM1-BD2-IN-8（0-100 μM；48小时）抑制了依赖PBRM1的前列腺癌细胞的生长[1]。

存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year

溶解度: DMSO : 55 mg/mL (173.4 mM)


关键字: PBRM1BD2IN8 | PBRM1-BD2-IN-8

相关产品: MI-3 | GSK1379725A | SR-0813 | Menin-MLL inhibitor 20 | SRX3177 | (+)-JQ1 PA | PROTAC BRD4 Degrader-3 | TP-472 | SMD-3040 | MG 149

相关库: Anti-Cancer Compound Library | Bioactive Compounds Library Max | Inhibitor Library | Epigenetics Compound Library | Anti-Cancer Active Compound Library | PPI Inhibitor Library | Histone Modification Compound Library | Bioactive Compound Library