Product Introduction
Bioactivity


英文名: GX 201

描述: GX 201 是选择性的 NaV1.7 抑制剂，其对 hNaV1.7 的 IC50 值为 <3.2 nM。

体内活性: GX 201在小鼠体内具有相对较长的半衰期。在自由血浆浓度大约是高亲和力通道阻断IC50的3倍时，GX 201能产生镇痛效果。GX 201抑制了由甲醛诱导的伤害感受反应以及由完全弗氏佐剂(CFA)引起的炎症性疼痛[1]。

存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year

溶解度: DMSO : 60 mg/mL (106.6 mM)


关键字: GX 201 | GX201

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相关库: Anti-Cancer Compound Library | Membrane Protein-targeted Compound Library | Bioactive Compounds Library Max | Inhibitor Library | Bioactive Compound Library