Product Introduction
Bioactivity


英文名: Transcrocetinate disodium

描述: Transcrocetinate disodium (Disodium trans-crocetinate) 从藏红花中提取的一种天然产物，是高亲和力NMDA 受体拮抗剂。

体外活性: Transcrocetinate表现出强烈的NMDA受体亲和力，被认为是藏红花中心神经系统(CNS)活性的主要因素。在10 μM浓度时，Transcrocetinate不影响细胞活性；然而，较高浓度(40-160 μM)则显著降低了细胞活性。

存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year

溶解度: H2O : 4.42 mg/mL (11.88 mM)
DMSO : Insoluble


关键字: Transcrocetinate | iGluR | Inhibitor | inhibit | Transcrocetinate disodium | Ionotropic glutamate receptors

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