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BIO-8169 是白细胞介素受体相关激酶 4 (IRAK 4) 的选择性抑制剂,IC50 为 0.23 nM。BIO-8169 在小鼠模型中表现出良好的药代动力学特征,减少促炎细胞因子的产生,并减轻 EAE 小鼠自身免疫性脑脊髓炎。BIO-
Oxygen Sensing Compound Library | 氧感应化合物库 | MedChemExpress (MCE)
Nucleotide Compound Library | 核苷类化合物库 | MedChemExpress (MCE)
Lipid Compound Library | 脂类化合物库 | MedChemExpress (MCE)
Glycoside Compound Library | 糖苷类化合物库 | MedChemExpress (MCE)
Macrocyclic Compound Library | 大环类化合物库 | MedChemExpress (MCE)
Anti-diabetic Compound Library | 抗糖尿病化合物库 | MedChemExpress (MCE)
Reprogramming Compound Library | 细胞重编程化合物库 | MedChemExpress (MCE)
Differentiation Inducing Compound Library | 诱导分化化合物库 | MedChemExpress (MCE)
Antioxidant Compound Library | 抗氧化化合物库 | MedChemExpress (MCE)
Covalent Screening Library Plus | 共价化合物库 Plus | MedChemExpress (MCE)