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GAT2711 (compound 3h) 是 α9 nAChR 的完全激动剂,EC50 为 230 nM。GAT2711 抑制了 THP-1 细胞中 ATP 诱导的 IL-1β 释放,在 α7 基因敲除小鼠中表现出镇痛活性。更多详情参考:h
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Levoglucosan-d7 | MedChemExpress (MCE)
1-Methylhistamine-d3 dihydrochloride | MedChemExpress (MCE)
Erythromycylamine-13C,d3 | 红霉胺-13C,d3 | MedChemExpress (MCE)
5-Methyl-5H-dibenzo[b,d]thiophen-5-ium trifluoromethanesulfonate-d3 | MedChemExpress (MCE)
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