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G-5758 是具有口服有效性的 IRE1α 抑制剂,对 XBP1s 的 IC50 为 38 nM。G-5758 可用于多发性骨髓瘤模型 (KMS-11) 的研究,大鼠口服剂量高达 500 mg/kg 时的耐受性仍然良好。G-5758 表现出
BCAM Human Pre-designed siRNA Set A | MedChemExpress (MCE)
BBX Human Pre-designed siRNA Set A | MedChemExpress (MCE)
BBS9 Human Pre-designed siRNA Set A | MedChemExpress (MCE)
BBS7 Human Pre-designed siRNA Set A | MedChemExpress (MCE)
BBS5 Human Pre-designed siRNA Set A | MedChemExpress (MCE)
BBS4 Human Pre-designed siRNA Set A | MedChemExpress (MCE)
BBS2 Human Pre-designed siRNA Set A | MedChemExpress (MCE)
BBS12 Human Pre-designed siRNA Set A | MedChemExpress (MCE)
BBS10 Human Pre-designed siRNA Set A | MedChemExpress (MCE)
BBS1 Human Pre-designed siRNA Set A | MedChemExpress (MCE)